Evigrade
Moderate

atorvastatin × omeprazole

HMG-CoA reductase inhibitors (statins)×Proton pump inhibitors

Mechanism

Omeprazole weakly inhibits CYP3A4 – atorvastatin exposure rises modestly (10–20 %). Clinically meaningful additional myopathy is rare.

Management

Routine dose adjustment is not required. If muscle pain develops, check CK and reconsider the statin.

Sources

All interactions

atorvastatin and omeprazole: interaction, management, sources – Evigrade